Table 1.
Enzyme selectivity profile of TAK-960 on selected kinases
Kinase
% inhibition at 1,000 nmol/L
IC
50
(nmol/L)
PLK1
101.6
0.8
PLK2
88
16.9
PLK3
81.8
50.2
FAK/PTK2
98.4
19.6
MLCK/MYLK
90.3
25.6
FES/FPS
81.5
58.2
282 kinases
<80