Table 1.

Quercetagetin is a selective inhibitor of the PIM1 kinase over other BAD(S112) kinases

KinaseIC50 (μmol/L)Log IC50 (μmol/L)SE of log IC50R2
PIM10.34−0.460.120.98
PIM23.450.550.220.94
PKA21.21.330.230.94
RSK22.820.450.090.99
  • NOTE: All data were derived from nonlinear regression analyses using a three-parameter logistic that assumes a Hill coefficient of −1.